Du, XiaochenHuang, JianjunNechaev, Anton A.Yao, RuweiGong, JingVan der Eycken, Erik V.Pereshivko, Olga P.Peshkov, Vsevolod A.2020-03-312020-03-312018-10-04Du, X.; Huang, J.; Nechaev, A. A.; Yao, R.; Gong, J.; Van der Eycken, E. V.; Pereshivko, O. P.; Peshkov, V. A. Beilstein J. Org. Chem. 2018, 14, 2572–2579. doi:10.3762/bjoc.14.234http://nur.nu.edu.kz/handle/123456789/4571A series of propargylamides containing an electron-rich benzene ring was prepared through the Ugi reaction of 3,5-dimethoxyaniline with various propiolic acids, aldehydes and isocyanides. Subjecting these adducts to a gold-catalyzed intramolecular alkyne hydroarylation process allowed to efficiently construct the 2-quinolone core bearing a branched substituent on the nitrogen atom...enAttribution-NonCommercial-ShareAlike 3.0 United Statesgold catalysishydroarylationUgi reactionArticle